adenosine antagonist-1 — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T10248	Adenosine antagonist-1		Adenosine Receptor
	Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.		Adenosine Receptor
T40307	Adenosine receptor antagonist 1
	Adenosine receptor antagonist 1 is a highly selective antagonist for the A2aR adenosine receptor, exhibiting an IC50 value of 0.29 nM. It demonstrates a remarkable 14-fold selectivity towards the A2aR receptor in compari...
T37792	A2A receptor antagonist 1	CPI-444 analog,A2A receptor antagonist 1	Adenosine Receptor
	A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.		Adenosine Receptor
T10058	A2B receptor antagonist 1		Adenosine Receptor
	A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.		Adenosine Receptor
T8312	Derenofylline		Adenosine Receptor
	Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)		Adenosine Receptor
T15418	GS-6201	CVT-6883	Adenosine Receptor
	GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors with a Ki of 22 nM.		Adenosine Receptor
T14078	AB928		Adenosine Receptor
	AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].		Adenosine Receptor
T22031	ANR 94		Adenosine Receptor
	ANR94 is a potent, selective antagonist of the adenosine A2A receptor (AA2AR), exhibiting a K_i value of 46 nM for the human AA2AR (hAA2AR). This compound shows promise for research into Parkinson's disease. [1] [2]		Adenosine Receptor
T70648	FK-352
	FK-352 is a pyrazolopyridine derivative and adenosine-1 receptor antagonist.
T24384	L-97-1	L97-1,L 97-1
	L-97-1 is an antagonist of the adenosine A1 receptor.
T62611	Adenosine receptor antagonist 2
	Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.
T70996	FK-838
	FK-838 is an adenosine subtype-1 receptor antagonist.
T60872	Adenosine receptor antagonist 3
	Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].
T72000	N 0840
	N 0840 is a selective, orally active A(1) adenosine receptor antagonist.
T61850	Adenosine receptor inhibitor 1
	Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >100...
T60580	A1AR antagonist 2
	A1AR antagonist 2 (compound 18h) is a potent antagonist of the A1 adenosine receptor (AR). A1AR antagonist 2 has Ki values of 1.49, 10.2, and 50.1 nM for hA 1, hA 2A, and hA 2B, respectively [1].
T62134	A1/A3 AR antagonist 1
	A1/A3 AR antagonist 1 (Compound 10) is a potent, dual adenosine 1 (A1) and adenosine 3 (A3) receptor antagonist that acts on human A1 (Ki: 37.6 nM), human A3 (Ki: 25.4 nM) and rat A1 (Ki: 1.47 nM). 1 Can be used to study...
T61536	A1AR antagonist 4
	A1AR antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the A1 adenosine receptor (A1AR). It possesses a pIC50 value of 5.51 and a pKi value of 6.29 [1].
T60687	A1AR antagonist 1
	A1AR antagonist 1 (compound 18g) is a potent antagonist of A1 adenosine receptor (AR). A1AR antagonist 1 has Ki values of 2.08, 6.91, and 31.2 nM for hA1, hA2A and hA2B, respectively [1].
T60615	A1AR antagonist 6
	A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].